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sc-PDB

An Annotated Database of Druggable Binding Sites from the Protein DataBank

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Distribution of Binding site similarity measured by Shaper
You can zoom onto the graph by using the mouse to make a selection

Binding Sites are compared using Shaper.
For more information, please see the following publication: Desaphy J. et al. Comparison and Druggability Prediction of protein-Ligand Binding sites from pharmacophore-annotated cavity shapes J. Chem. Inf. Model., 2012, 52(8), pp2287-2299
Binding Sites are considered as similar when the similarity value is greater than 0.44

Reference Protein Data Bank Entry :
PDB IDHETUniprot NameEC Number
3bzuA21Corticosteroid 11-beta-dehydrogenase isozyme 11.1.1.146

Complex with similar binding sites

PDB ID HET Uniprot Name EC Number Binding Site
Similarity
Align
3bzuA21Corticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1461.000
3byzH11Corticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.612
3oq13OQCorticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.606
3fcoIIGCorticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.592
3d3eD3ECorticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.585
2iltNN1Corticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.572
3czr3CZCorticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.569
3h6k33TCorticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.564
4bb5HD2Corticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.563
1xu9CPSCorticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.560
3ch6311Corticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.553
3gmd2M3Corticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.543
4bb6HD1Corticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.541
3vrwYS5Vitamin D3 receptor/0.531
3tfq07MCorticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.530
4hfr14MCorticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.526
3g493G4Corticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.518
3d5qT30Corticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.512
1xu7CPSCorticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.506
3ey4352Corticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.497
1y5rC0RCorticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.493
4g1z0VPVitamin D3 receptor A/0.493
3c0g3AMPeripheral plasma membrane protein CASK2.7.11.10.486
1kvoOAPPhospholipase A2, membrane associated/0.484
2zl9VDAVitamin D3 receptor/0.484
3vt5YI2Vitamin D3 receptor/0.483
3l0lHC3Nuclear receptor ROR-gamma/0.482
3gytDL4Nuclear hormone receptor of the steroid/thyroid hormone receptors superfamily/0.480
3p9tTCLRepressor/0.478
2hamC33Vitamin D3 receptor/0.475
4g1d0VKVitamin D3 receptor A/0.475
1cqp803Integrin alpha-L/0.474
2hb8MVDVitamin D3 receptor/0.474
3vt65YIVitamin D3 receptor/0.473
2qo5CHDFatty acid-binding protein 10-A, liver basic/0.472
1s19MC9Vitamin D3 receptor/0.471
2rbeZMGCorticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.471
4jbtASDCytochrome P450 monooxygenase/0.471
3w0aDS5Vitamin D3 receptor/0.470
4lb2DM5Serum albumin/0.470
4r20AERCytochrome P450 family 17 polypeptide 2/0.470
1ie8KH1Vitamin D3 receptor/0.469
2po7CHDFerrochelatase, mitochondrial4.99.1.10.469
4nky3QZSteroid 17-alpha-hydroxylase/17,20 lyase/0.469
1fm7DFVChalcone--flavonone isomerase 15.5.1.60.468
3w5p4OAVitamin D3 receptor/0.468
4ia2BIVVitamin D3 receptor A/0.467
3kytHC2Nuclear receptor ROR-gamma/0.466
3up3XCAaceDAF-12/0.466
3vrvYSDVitamin D3 receptor/0.466
4j6dTESCytochrome P450 monooxygenase/0.466
2qd4CHDFerrochelatase, mitochondrial4.99.1.10.464
3vtbTKAVitamin D3 receptor/0.464
4ia7BIVVitamin D3 receptor A/0.464
1tbbROLcAMP-specific 3',5'-cyclic phosphodiesterase 4D3.1.4.530.463
1zx1CB1Ribosyldihydronicotinamide dehydrogenase [quinone]/0.463
3vtcTK3Vitamin D3 receptor/0.463
4jib1L6cGMP-dependent 3',5'-cyclic phosphodiesterase3.1.4.170.463
1e7aPFLSerum albumin/0.462
1rkhVD2Vitamin D3 receptor/0.462
2zevB71Geranylgeranyl pyrophosphate synthase/0.462
2zlcVDXVitamin D3 receptor/0.462
3vt9YI4Vitamin D3 receptor/0.462
3w1wCHDFerrochelatase, mitochondrial4.99.1.10.462
4g210VPVitamin D3 receptor A/0.462
4g95OAGDihydrofolate reductase1.5.1.30.462
4nb6444Nuclear receptor ROR-gamma/0.462
1kk4ACOStreptogramin A acetyltransferase2.3.10.461
1rdtL79Retinoic acid receptor RXR-alpha/0.461
3w5rLOAVitamin D3 receptor/0.461
4bb3KKAIsopenicillin N synthase1.21.3.10.461
4ez8DHFThymidylate synthase2.1.1.450.461
4g20484Vitamin D3 receptor A/0.461
4jlj1NMDeoxycytidine kinase2.7.1.740.461
4q0a4OAVitamin D3 receptor A/0.461
1txiTX5Vitamin D3 receptor/0.460
2harOCCVitamin D3 receptor/0.460
3vrtYS2Vitamin D3 receptor/0.460
4nkvAERSteroid 17-alpha-hydroxylase/17,20 lyase/0.459
1iyzNDPProbable quinone oxidoreductase/0.458
2hc4VDXVitamin D3 receptor A/0.458
2zlaVDBVitamin D3 receptor/0.458
3ox1695Ribosyldihydronicotinamide dehydrogenase [quinone]/0.458
3vt3VDXVitamin D3 receptor/0.458
3w0gW07Vitamin D3 receptor/0.458
1felFENRetinol-binding protein 4/0.457
1ndzFR5Adenosine deaminase3.5.4.40.457
2aibERGBeta-elicitin cinnamomin/0.457
2g2hP16Tyrosine-protein kinase ABL12.7.10.20.457
4o701QKBromodomain-containing protein 4/0.457
1db48INPhospholipase A2, membrane associated/0.456
2hrcCHDFerrochelatase, mitochondrial4.99.1.10.456
2o4jVD4Vitamin D3 receptor/0.456
3uic09TEnoyl-[acyl-carrier-protein] reductase [NADH]/0.456
4ia1BIVVitamin D3 receptor A/0.456
1db1VDXVitamin D3 receptor/0.455
3dr1C5DVitamin D3 receptor A/0.455
3g8eIS1Nicotinamide phosphoribosyltransferase2.4.2.120.455
1dnaCB3Thymidylate synthase/0.454
1s0zEB1Vitamin D3 receptor/0.454
1x8lOXRRetinol dehydratase/0.454
2jg7NADAntiquitin/0.454
2y60M8FIsopenicillin N synthase1.21.3.10.454
3v4eCOAPutative acetyltransferase SACOL25702.3.10.454
3w0iO11Vitamin D3 receptor/0.454
4bvaT3Ketimine reductase mu-crystallin1.5.1.250.454
4h9614QDihydrofolate reductase1.5.1.30.454
3reyXACAdenosine receptor A2a/0.454
1eioGCHGastrotropin/0.453
1ie9VDXVitamin D3 receptor/0.453
1l2jETCEstrogen receptor beta/0.453
1zeoC01Peroxisome proliferator-activated receptor gamma/0.453
3h18PMSEsterase/lipase/0.453
3vt45YIVitamin D3 receptor/0.453
3w0hW12Vitamin D3 receptor/0.453
3w5q3KLVitamin D3 receptor/0.453
4e37NDPCatalase1.11.1.60.453
4eh6IRGMitogen-activated protein kinase 14/0.453
4fhh0U3Vitamin D3 receptor A/0.453
4g1y0VOVitamin D3 receptor A/0.453
4iaq2GM5-hydroxytryptamine receptor 1B/0.453
4jvmXDIEstrogen sulfotransferase2.8.2.40.453
4wa9AXITyrosine-protein kinase ABL12.7.10.20.453
1db56INPhospholipase A2, membrane associated/0.452
1fmjRTLRetinol dehydratase/0.452
1kquBR4Phospholipase A2, membrane associated/0.452
1xddAAYIntegrin alpha-L/0.452
2hw2RFPRifampin ADP-ribosyl transferase/0.452
3a783EVVitamin D3 receptor/0.452
3gyuDL7Nuclear hormone receptor of the steroid/thyroid hormone receptors superfamily/0.452
4g2h0VQVitamin D3 receptor A/0.452
1d3hA26Dihydroorotate dehydrogenase (quinone), mitochondrial1.3.5.20.451
1ep4S11Gag-Pol polyprotein2.7.7.490.451
1re9DSOCamphor 5-monooxygenase1.14.15.10.451
1rk3VDXVitamin D3 receptor/0.451
1uzwCDHIsopenicillin N synthase1.21.3.10.451
2xlsFADPutative flavin-containing monooxygenase/0.451
2z3uCRRCytochrome P450/0.451
3p99LNPLanosterol 14-alpha-demethylase/0.451
3qm4PN0Cytochrome P450 2D6/0.451
4i9i1DYTankyrase-12.4.2.300.451
4yt5H4MH(2)-forming methylenetetrahydromethanopterin dehydrogenase-related protein MJ1338/0.451
1mvtDTMDihydrofolate reductase1.5.1.30.450
1tvrTB9Gag-Pol polyprotein2.7.7.490.450
2bu9HFVIsopenicillin N synthase1.21.3.10.450
2fr0NDP6-deoxyerythronolide-B synthase EryA1, modules 1 and 2/0.450
2hb7O1CVitamin D3 receptor/0.450
4jvb1M0Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta/0.450
1lriCLRBeta-elicitin cryptogein/0.449
1lwlDSOCamphor 5-monooxygenase1.14.15.10.449
1rjkVDZVitamin D3 receptor/0.449
2fb8215Serine/threonine-protein kinase B-raf2.7.11.10.449
2hasC3OVitamin D3 receptor/0.449
3d75NBBPheromone-binding protein ASP1/0.449
3gkjHC3Niemann-Pick C1 protein/0.449
3kpzZNEVitamin D3 receptor/0.449
3v94WYQPhosphodiesterase/0.449
3w5tLHPVitamin D3 receptor/0.449
4l8u9AZSerum albumin/0.449
4l9q9TPSerum albumin/0.449
4rujVDXVitamin D3 receptor A/0.449
4xivACPChemotaxis protein CheA2.7.13.30.449
5cp8TCUEnoyl-[acyl-carrier-protein] reductase [NADH]1.3.1.90.449
1m52P17Tyrosine-protein kinase ABL12.7.10.20.448
2xk85R1Serine/threonine-protein kinase Nek22.7.11.10.448
4biiPYWEnoyl-[acyl-carrier-protein] reductase [NADH]1.3.1.90.448
4iteTEYVitamin D3 receptor/0.448
4j6bPLOCytochrome P450 monooxygenase/0.448
5k2aZMAAdenosine receptor A2a/0.448
1iolESTEstradiol 17-beta-dehydrogenase 11.1.1.620.447
1kb9SMACytochrome b/0.447
2o4rVD5Vitamin D3 receptor/0.447
2vagV25Dual specificity protein kinase CLK12.7.12.10.447
3a1l2CCCytochrome P450/0.447
3adaNADSubunit alpha of sarocosine oxidase/0.447
3pqbVGPPutative oxidoreductase/0.447
3tm5SFGUncharacterized protein/0.447
3w0jT08Vitamin D3 receptor/0.447
4eevL1XHepatocyte growth factor receptor2.7.10.10.447
4jlk1NODeoxycytidine kinase2.7.1.740.447
4oztP1AEcdysone receptor, putative/0.447
4rupH97Vitamin D3 receptor A/0.447
1p44GEQEnoyl-[acyl-carrier-protein] reductase [NADH]1.3.1.90.446
1y60H4M5,6,7,8-tetrahydromethanopterin hydro-lyase4.2.1.1470.446
2b01TUDPhospholipase A2, major isoenzyme3.1.1.40.446
2b365PPEnoyl-[acyl-carrier-protein] reductase [NADH]1.3.1.90.446
2jdvL20cAMP-dependent protein kinase catalytic subunit alpha2.7.11.110.446
3acw651Dehydrosqualene synthase/0.446
3fnhJPJEnoyl-[acyl-carrier-protein] reductase [NADH]1.3.1.90.446
3p3zP3ZPutative cytochrome P450/0.446
3p6oETGCamphor 5-monooxygenase1.14.15.10.446
3zlmANPAdenosine monophosphate-protein transferase NmFic2.7.7.n10.446
3pwhZMAAdenosine receptor A2a/0.446
1m7aMQUDihydrofolate reductase1.5.1.30.445
1rkgVD1Vitamin D3 receptor/0.445
1xoqROFcAMP-specific 3',5'-cyclic phosphodiesterase 4D3.1.4.530.445
2aazCB3Thymidylate synthase2.1.1.450.445
2xk4OL2Serine/threonine-protein kinase Nek22.7.11.10.445
3lu8IQXSerum albumin/0.445
3o73O73Ribosyldihydronicotinamide dehydrogenase [quinone]/0.445
3sqwANPATP-dependent RNA helicase MSS116, mitochondrial3.6.4.130.445
4e5yNDPGDP-L-fucose synthase1.1.1.2710.445
4m6p20RNicotinamide phosphoribosyltransferase2.4.2.120.445
4y8vADPAcyl-CoA synthetase (NDP forming)/0.445
2wufKEM4,5:9,10-diseco-3-hydroxy-5,9,17-trioxoandrosta-1(10),2-diene-4-oate hydrolase3.7.1.170.444
2y6fM9FIsopenicillin N synthase1.21.3.10.444
3abaFLICytochrome P450/0.444
3h3sH15Collagen type IV alpha-3-binding protein/0.444
3r04UNQSerine/threonine-protein kinase pim-12.7.11.10.444
3vtdTKDVitamin D3 receptor/0.444
4oj4DIFPeroxisome proliferator-activated receptor gamma/0.444
5k2bZMAAdenosine receptor A2a/0.444
1dcyI3NPhospholipase A2, membrane associated/0.443
1n4hREANuclear receptor ROR-beta/0.443
3c1tMYCDihydroflavonol 4-reductase1.1.1.2190.443
3el8PD5Proto-oncogene tyrosine-protein kinase Src2.7.10.20.443
3lkhLT6Genome polyprotein2.7.7.480.443
3nrrD16Bifunctional dihydrofolate reductase-thymidylate synthase/0.443
3p6nDSOCamphor 5-monooxygenase1.14.15.10.443
3pm1ETHTH-type transcriptional regulator QacR/0.443
3t8xT8XT-cell surface glycoprotein CD1b/0.443
4h9506UDihydrofolate reductase1.5.1.30.443
4lwwLWWNicotinamide phosphoribosyltransferase2.4.2.120.443
4nieNBHNuclear receptor ROR-gamma/0.443
4x5gFOLDihydrofolate reductase1.5.1.30.443
5jtbZMAAdenosine receptor A2a/0.443
1dajMOTDihydrofolate reductase1.5.1.30.442
1fduESTEstradiol 17-beta-dehydrogenase 11.1.1.620.442
1fm4DXCMajor pollen allergen Bet v 1-L/0.442
1hvyD16Thymidylate synthase2.1.1.450.442
1o6rR19Squalene--hopene cyclase4.2.1.1290.442
2hcdBIVVitamin D3 receptor A/0.442
2p1u4TNRetinoic acid receptor RXR-alpha/0.442
2w0bCMWLanosterol 14-alpha demethylase1.14.13.700.442
2w4qCBWProstaglandin reductase 21.3.1.480.442
2y30SM8Putative repressor SimReg2/0.442
3dokGWJPol protein/0.442
3h1jSMACytochrome b/0.442
3oafOAGDihydrofolate reductase1.5.1.30.442
3vsoEK1Peroxisome proliferator-activated receptor gamma/0.442
4inb1F6Gag protein/0.442
4pkl1GHUncharacterized protein/0.442
5dozNDPJamJ/0.442
1ia3TQ5Dihydrofolate reductase1.5.1.30.441
1w06W05Isopenicillin N synthase1.21.3.10.441
2bikBI1Serine/threonine-protein kinase pim-12.7.11.10.441
2fzhDH1Dihydrofolate reductase1.5.1.30.441
2ibzSMACytochrome b/0.441
2jn3JN3Fatty acid-binding protein, liver/0.441
2pnjCHDFerrochelatase, mitochondrial4.99.1.10.441
3g70A5TRenin3.4.23.150.441
3hub469Mitogen-activated protein kinase 14/0.441
3ozd4CTS-methyl-5'-thioadenosine phosphorylase/0.441
3rm618ZCyclin-dependent kinase 22.7.11.220.441
3s41S41Glucokinase2.7.1.20.441
4fex0TOAminoglycoside 3'-phosphotransferase AphA1-IAB/0.441
4fhi0S4Vitamin D3 receptor A/0.441
4h9753SDihydrofolate reductase1.5.1.30.441
4ruoBIVVitamin D3 receptor A/0.441
5dq8FLFTranscriptional enhancer factor TEF-4/0.441
5uviZMAAdenosine receptor A2a/0.441
4k5y1Q5Corticotropin-releasing factor receptor 1/0.441
1dkfBMSRetinoic acid receptor alpha/0.440
1nq7ARLNuclear receptor ROR-beta/0.440
1osvCHCBile acid receptor/0.440
1qxlFR8Adenosine deaminase3.5.4.40.440
2ban357Gag-Pol polyprotein2.7.7.490.440
2vqoTFGHistone deacetylase 43.5.1.980.440
2y98MIVMycinamicin IV hydroxylase/epoxidase/0.440
3ctj320Hepatocyte growth factor receptor2.7.10.10.440
3l08ZIGPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform2.7.1.1530.440
3lz6A0DCorticosteroid 11-beta-dehydrogenase isozyme 11.1.1.1460.440
3vruYS3Vitamin D3 receptor/0.440
3vt8YI3Vitamin D3 receptor/0.440
4a322CDGlycylpeptide N-tetradecanoyltransferase/0.440
4cax646Glycylpeptide N-tetradecanoyltransferase2.3.1.970.440
4itfTFYVitamin D3 receptor/0.440
4rlh0WEEnoyl-[acyl-carrier-protein] reductase [NADH]/0.440
5hs1VORLanosterol 14-alpha demethylase/0.440